It is our great honor to organize “The 3rd International Symposium on Natural Product Synthesis and Process Methods for Drug Manufacture (NPSPM)” in Beijing, China, from Oct 14 (Friday) to 16 (Sunday), 2016. This symposium will focus on the frontiers of natural product synthesis and discovery and develoment of novel reactions and process methods towards drug manufacture. Twenty-six world-famous academic scholars and industrial scientists from various countries and regions have accepted our invitations and will deliver their plenary and invited talks during the symposium. Selected posters will also be presented to further enrich this symposium. We welcome all of you to Beijing to enjoy this symposium and the beautiful organic chemistry presented.